Compile Data Set for Download or QSAR

Found 90 hits of kd data for polymerid = 3688   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199423 (CHEMBL3983476) Show SMILES COc1nn2cc(nc2s1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-2-4-8(12)5-3-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	621	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199423 (CHEMBL3983476) Show SMILES COc1nn2cc(nc2s1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-2-4-8(12)5-3-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	621	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced P-selectin activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199414 (CHEMBL3968857) Show SMILES COc1nn2cc(nc2s1)-c1cccc(F)c1 Show InChI InChI=1S/C11H8FN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-3-2-4-8(12)5-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	675	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199414 (CHEMBL3968857) Show SMILES COc1nn2cc(nc2s1)-c1cccc(F)c1 Show InChI InChI=1S/C11H8FN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-3-2-4-8(12)5-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	676	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199436 (CHEMBL3947023) Show SMILES COc1nn2cc(nc2s1)-c1ccccc1 Show InChI InChI=1S/C11H9N3OS/c1-15-11-13-14-7-9(12-10(14)16-11)8-5-3-2-4-6-8/h2-7H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	757	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199436 (CHEMBL3947023) Show SMILES COc1nn2cc(nc2s1)-c1ccccc1 Show InChI InChI=1S/C11H9N3OS/c1-15-11-13-14-7-9(12-10(14)16-11)8-5-3-2-4-6-8/h2-7H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	759	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199434 (CHEMBL3975497) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)C#N Show InChI InChI=1S/C12H8N4OS/c1-17-12-15-16-7-10(14-11(16)18-12)9-4-2-8(6-13)3-5-9/h2-5,7H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	933	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199434 (CHEMBL3975497) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)C#N Show InChI InChI=1S/C12H8N4OS/c1-17-12-15-16-7-10(14-11(16)18-12)9-4-2-8(6-13)3-5-9/h2-5,7H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	937	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199420 (CHEMBL3933579) Show SMILES COc1nn2cc(nc2s1)-c1cc2cc(OC(F)(F)F)ccc2n1C Show InChI InChI=1S/C15H11F3N4O2S/c1-21-11-4-3-9(24-15(16,17)18)5-8(11)6-12(21)10-7-22-13(19-10)25-14(20-22)23-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	977	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199420 (CHEMBL3933579) Show SMILES COc1nn2cc(nc2s1)-c1cc2cc(OC(F)(F)F)ccc2n1C Show InChI InChI=1S/C15H11F3N4O2S/c1-21-11-4-3-9(24-15(16,17)18)5-8(11)6-12(21)10-7-22-13(19-10)25-14(20-22)23-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced P-selectin activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199420 (CHEMBL3933579) Show SMILES COc1nn2cc(nc2s1)-c1cc2cc(OC(F)(F)F)ccc2n1C Show InChI InChI=1S/C15H11F3N4O2S/c1-21-11-4-3-9(24-15(16,17)18)5-8(11)6-12(21)10-7-22-13(19-10)25-14(20-22)23-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced P-selectin activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199420 (CHEMBL3933579) Show SMILES COc1nn2cc(nc2s1)-c1cc2cc(OC(F)(F)F)ccc2n1C Show InChI InChI=1S/C15H11F3N4O2S/c1-21-11-4-3-9(24-15(16,17)18)5-8(11)6-12(21)10-7-22-13(19-10)25-14(20-22)23-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199433 (CHEMBL3902806) Show SMILES COc1nn2cc(nc2s1)-c1ccc(F)c(c1)C(F)(F)F Show InChI InChI=1S/C12H7F4N3OS/c1-20-11-18-19-5-9(17-10(19)21-11)6-2-3-8(13)7(4-6)12(14,15)16/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.09E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199433 (CHEMBL3902806) Show SMILES COc1nn2cc(nc2s1)-c1ccc(F)c(c1)C(F)(F)F Show InChI InChI=1S/C12H7F4N3OS/c1-20-11-18-19-5-9(17-10(19)21-11)6-2-3-8(13)7(4-6)12(14,15)16/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199441 (CHEMBL3948984) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)S(C)(=O)=O Show InChI InChI=1S/C12H11N3O3S2/c1-18-12-14-15-7-10(13-11(15)19-12)8-3-5-9(6-4-8)20(2,16)17/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199441 (CHEMBL3948984) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)S(C)(=O)=O Show InChI InChI=1S/C12H11N3O3S2/c1-18-12-14-15-7-10(13-11(15)19-12)8-3-5-9(6-4-8)20(2,16)17/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199417 (CHEMBL3963226) Show SMILES COc1nn2cc(nc2s1)-c1c(F)cccc1F Show InChI InChI=1S/C11H7F2N3OS/c1-17-11-15-16-5-8(14-10(16)18-11)9-6(12)3-2-4-7(9)13/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.29E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199417 (CHEMBL3963226) Show SMILES COc1nn2cc(nc2s1)-c1c(F)cccc1F Show InChI InChI=1S/C11H7F2N3OS/c1-17-11-15-16-5-8(14-10(16)18-11)9-6(12)3-2-4-7(9)13/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199425 (CHEMBL3950308) Show SMILES COc1nn2cc(nc2s1)-c1cccc(c1)C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-3-2-4-8(5-7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.31E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199425 (CHEMBL3950308) Show SMILES COc1nn2cc(nc2s1)-c1cccc(c1)C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-3-2-4-8(5-7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.32E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199419 (CHEMBL3918711) Show SMILES COc1nn2cc(nc2s1)-c1ccccc1C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-4-2-3-5-8(7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.32E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199419 (CHEMBL3918711) Show SMILES COc1nn2cc(nc2s1)-c1ccccc1C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-4-2-3-5-8(7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.33E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199440 (CHEMBL3909608) Show SMILES COc1nn2cc(nc2s1)-c1ccc(Cl)c(Cl)c1 Show InChI InChI=1S/C11H7Cl2N3OS/c1-17-11-15-16-5-9(14-10(16)18-11)6-2-3-7(12)8(13)4-6/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.45E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199440 (CHEMBL3909608) Show SMILES COc1nn2cc(nc2s1)-c1ccc(Cl)c(Cl)c1 Show InChI InChI=1S/C11H7Cl2N3OS/c1-17-11-15-16-5-9(14-10(16)18-11)6-2-3-7(12)8(13)4-6/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.46E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199418 (CHEMBL3973767) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC(F)F)cc1 Show InChI InChI=1S/C12H9F2N3O2S/c1-18-12-16-17-6-9(15-11(17)20-12)7-2-4-8(5-3-7)19-10(13)14/h2-6,10H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	2.51E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199418 (CHEMBL3973767) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC(F)F)cc1 Show InChI InChI=1S/C12H9F2N3O2S/c1-18-12-16-17-6-9(15-11(17)20-12)7-2-4-8(5-3-7)19-10(13)14/h2-6,10H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	2.54E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199426 (CHEMBL3905565) Show SMILES CN(C)c1nn2cc(nc2s1)-c1c(F)cccc1F Show InChI InChI=1S/C12H10F2N4S/c1-17(2)12-16-18-6-9(15-11(18)19-12)10-7(13)4-3-5-8(10)14/h3-6H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199430 (CHEMBL3924666) Show SMILES COc1nn2cc(nc2s1)-c1ccccc1[N+]([O-])=O Show InChI InChI=1S/C11H8N4O3S/c1-18-11-13-14-6-8(12-10(14)19-11)7-4-2-3-5-9(7)15(16)17/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.79E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199430 (CHEMBL3924666) Show SMILES COc1nn2cc(nc2s1)-c1ccccc1[N+]([O-])=O Show InChI InChI=1S/C11H8N4O3S/c1-18-11-13-14-6-8(12-10(14)19-11)7-4-2-3-5-9(7)15(16)17/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.84E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199431 (CHEMBL3927486) Show SMILES COc1nn2cc(nc2s1)-c1cc(cc(c1)C(F)(F)F)C(F)(F)F Show InChI InChI=1S/C13H7F6N3OS/c1-23-11-21-22-5-9(20-10(22)24-11)6-2-7(12(14,15)16)4-8(3-6)13(17,18)19/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.62E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199431 (CHEMBL3927486) Show SMILES COc1nn2cc(nc2s1)-c1cc(cc(c1)C(F)(F)F)C(F)(F)F Show InChI InChI=1S/C13H7F6N3OS/c1-23-11-21-22-5-9(20-10(22)24-11)6-2-7(12(14,15)16)4-8(3-6)13(17,18)19/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.62E+3	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199415 (CHEMBL3906686) Show SMILES CNc1nn2cc(nc2s1)-c1c(F)cccc1F Show InChI InChI=1S/C11H8F2N4S/c1-14-10-16-17-5-8(15-11(17)18-10)9-6(12)3-2-4-7(9)13/h2-5H,1H3,(H,14,16)	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 1 (Homo sapiens (Human))	BDBM50199420 (CHEMBL3933579) Show SMILES COc1nn2cc(nc2s1)-c1cc2cc(OC(F)(F)F)ccc2n1C Show InChI InChI=1S/C15H11F3N4O2S/c1-21-11-4-3-9(24-15(16,17)18)5-8(11)6-12(21)10-7-22-13(19-10)25-14(20-22)23-2/h3-7H,1-2H3	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR1 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199429 (CHEMBL3896629) Show SMILES COc1nn2cc(nc2s1)-c1cccc(c1)[N+]([O-])=O Show InChI InChI=1S/C11H8N4O3S/c1-18-11-13-14-6-9(12-10(14)19-11)7-3-2-4-8(5-7)15(16)17/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199422 (CHEMBL3904669) Show SMILES COc1nn2cc(nc2s1)-c1ccc(O)cc1 Show InChI InChI=1S/C11H9N3O2S/c1-16-11-13-14-6-9(12-10(14)17-11)7-2-4-8(15)5-3-7/h2-6,15H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 1 (Homo sapiens (Human))	BDBM50199420 (CHEMBL3933579) Show SMILES COc1nn2cc(nc2s1)-c1cc2cc(OC(F)(F)F)ccc2n1C Show InChI InChI=1S/C15H11F3N4O2S/c1-21-11-4-3-9(24-15(16,17)18)5-8(11)6-12(21)10-7-22-13(19-10)25-14(20-22)23-2/h3-7H,1-2H3	PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR1 in human platelets assessed as inhibition of activating peptide-induced P-selectin activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199422 (CHEMBL3904669) Show SMILES COc1nn2cc(nc2s1)-c1ccc(O)cc1 Show InChI InChI=1S/C11H9N3O2S/c1-16-11-13-14-6-9(12-10(14)17-11)7-2-4-8(15)5-3-7/h2-6,15H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199428 (CHEMBL3890362) Show SMILES COc1nn2cc(nc2s1)-c1cccc(Cl)c1 Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-3-2-4-8(12)5-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199428 (CHEMBL3890362) Show SMILES COc1nn2cc(nc2s1)-c1cccc(Cl)c1 Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-3-2-4-8(12)5-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199429 (CHEMBL3896629) Show SMILES COc1nn2cc(nc2s1)-c1cccc(c1)[N+]([O-])=O Show InChI InChI=1S/C11H8N4O3S/c1-18-11-13-14-6-9(12-10(14)19-11)7-3-2-4-8(5-7)15(16)17/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair

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